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- (6aS)-1,10-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,9-diol
- 16-base single stranded RNA targeting miR-23b linked to oleic acid
- Humanised IgG1 kappa fragment antibody targeting TfR1 conjugated to P125 oligonucleotide
- Humanised IgG1 monoclonal antibody against TfR1 conjugated to double stranded siRNA oligonucleotide against DMPK via a non-cleavable linker